4-[1-[4-[2-(dimethylamino)ethoxy]phenyl]-2-phenylbut-1-enyl]phenol has been researched along with afimoxifene in 11 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 4 (36.36) | 18.7374 |
1990's | 1 (9.09) | 18.2507 |
2000's | 4 (36.36) | 29.6817 |
2010's | 2 (18.18) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bischoff, SF; Buhl, T; Floersheim, P; Fournier, B; Halleux, C; Kallen, J; Keller, H; Renaud, J; Schlaeppi, JM; Stark, W | 1 |
Chao, EY; Collins, JL; Gaillard, S; Jones, DG; McDonnell, DP; Miller, AB; Orband-Miller, LA; Shearer, BG; Willson, TM; Zuercher, WJ | 1 |
Chao, EY; Collins, JL; Gaillard, S; McDonnell, DP; Miller, AB; Nolte, RT; Orband-Miller, LA; Wang, L; Willson, TM; Zuercher, WJ | 1 |
Devleeschouwer, N; Foster, AB; Jarman, M; Leclercq, G; Leung, OT; McCague, R | 1 |
Bagley, JR; Mokler, CM; Ruenitz, PC | 1 |
Bignon, E; Crastes de Paulet, A; Doré, JC; Gilbert, J; Miquel, JF; Ojasoo, T; Pons, M; Raynaud, JP | 1 |
Abecassis, J; Bignon, E; Crastes de Paulet, AC; Doré, JC; Gilbert, J; Miquel, JF; Ojasoo, T; Pons, M; Raynaud, JP | 1 |
Jordan, VC; Leclercq, G; McCague, R | 1 |
Hillard, EA; Huché, M; Jaouen, G; Pigeon, P; Salomon, E; Top, S; Vessières, A | 1 |
Curpan, RF; Jordan, VC; Lewis-Wambi, JS; Maximov, PY; Myers, CB | 1 |
Forman, BM; Huss, JM; Li, H; Yu, DD | 1 |
11 other study(ies) available for 4-[1-[4-[2-(dimethylamino)ethoxy]phenyl]-2-phenylbut-1-enyl]phenol and afimoxifene
Article | Year |
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Estrogen receptor modulators: identification and structure-activity relationships of potent ERalpha-selective tetrahydroisoquinoline ligands.
Topics: Administration, Oral; Animals; Binding Sites; Biological Availability; Cell Division; Crystallography, X-Ray; Estradiol; Estrogen Receptor alpha; Estrogen Receptor beta; Estrogen Receptor Modulators; Female; HeLa Cells; Humans; Isoquinolines; Ligands; Models, Molecular; Radioligand Assay; Raloxifene Hydrochloride; Rats; Receptors, Estrogen; Stereoisomerism; Structure-Activity Relationship; Transcription, Genetic; Tumor Cells, Cultured | 2003 |
Identification and structure-activity relationship of phenolic acyl hydrazones as selective agonists for the estrogen-related orphan nuclear receptors ERRbeta and ERRgamma.
Topics: Binding, Competitive; Estrogen Receptor beta; Fluorescence Resonance Energy Transfer; Genes, Reporter; Heat-Shock Proteins; HeLa Cells; Humans; Hydrazines; Ligands; Molecular Mimicry; Peroxisome Proliferator-Activated Receptor Gamma Coactivator 1-alpha; Phenols; Receptors, Estrogen; Structure-Activity Relationship; Transcription Factors | 2005 |
Structure-guided synthesis of tamoxifen analogs with improved selectivity for the orphan ERRgamma.
Topics: Binding Sites; Crystallography, X-Ray; Drug Design; Estrogen Receptor alpha; Humans; Ligands; Models, Molecular; Molecular Structure; Receptors, Cytoplasmic and Nuclear; Receptors, Estrogen; Structure-Activity Relationship; Tamoxifen | 2006 |
Hydroxy derivatives of tamoxifen.
Topics: Binding, Competitive; Breast Neoplasms; Cell Division; Cell Line; Chemical Phenomena; Chemistry; Female; Humans; Hydroxylation; Receptors, Estrogen; Stereoisomerism; Structure-Activity Relationship; Tamoxifen | 1985 |
Estrogenic and antiestrogenic activity of monophenolic analogues of tamoxifen, (Z)-2-[p-(1,2-diphenyl-1-butenyl)phenoxy]-N, N-dimethylethylamine.
Topics: Animals; Chemical Phenomena; Chemistry; Cytosol; Drug Stability; Estrogen Antagonists; Estrogens; Female; In Vitro Techniques; Magnetic Resonance Spectroscopy; Organ Size; Rats; Rats, Inbred Strains; Receptors, Estrogen; Tamoxifen; Uterus | 1982 |
Multivariate analysis by the minimum spanning tree method of the structural determinants of diphenylethylenes and triphenylacrylonitriles implicated in estrogen receptor binding, protein kinase C activity, and MCF7 cell proliferation.
Topics: Acrylonitrile; Animals; Antineoplastic Agents; Breast Neoplasms; Cell Division; Dose-Response Relationship, Drug; Estrogen Antagonists; Female; Humans; Multivariate Analysis; Protein Kinase C; Rats; Receptors, Estrogen; Stilbenes; Structure-Activity Relationship; Tumor Cells, Cultured | 1992 |
Effect of triphenylacrylonitrile derivatives on estradiol-receptor binding and on human breast cancer cell growth.
Topics: Animals; Breast Neoplasms; Cattle; Cell Division; Cell Line; Chemical Phenomena; Chemistry; Cytosol; Female; Growth Inhibitors; Humans; Isomerism; Mice; Nitriles; Rats; Receptors, Estradiol; Structure-Activity Relationship; Terphenyl Compounds; Tumor Cells, Cultured | 1989 |
Nonisomerizable analogues of (Z)- and (E)-4-hydroxytamoxifen. Synthesis and endocrinological properties of substituted diphenylbenzocycloheptenes.
Topics: Animals; Benzocycloheptenes; Breast Neoplasms; Cell Division; Chemical Phenomena; Chemistry; Female; Humans; Organ Size; Rats; Rats, Inbred Strains; Receptors, Estrogen; Tamoxifen; Tumor Cells, Cultured; Uterus | 1988 |
Selective estrogen receptor modulators in the ruthenocene series. Synthesis and biological behavior.
Topics: Antineoplastic Agents; Breast Neoplasms; Cell Line, Tumor; Cell Proliferation; Drug Screening Assays, Antitumor; Electrochemistry; Estrogen Receptor alpha; Estrogen Receptor beta; Estrogen Receptor Modulators; Female; Humans; Models, Molecular; Neoplasms, Hormone-Dependent; Organometallic Compounds; Ruthenium; Stereoisomerism; Structure-Activity Relationship; Tamoxifen | 2005 |
Structure-function relationships of estrogenic triphenylethylenes related to endoxifen and 4-hydroxytamoxifen.
Topics: Binding Sites; Breast Neoplasms; Cell Line, Tumor; Cell Proliferation; Crystallography, X-Ray; Estrogen Antagonists; Estrogens, Non-Steroidal; Ethylenes; Female; Humans; Models, Molecular; Receptors, Estrogen; Stereoisomerism; Structure-Activity Relationship; Tamoxifen | 2010 |
Identification of novel inverse agonists of estrogen-related receptors ERRγ and ERRβ.
Topics: Crystallography, X-Ray; Drug Inverse Agonism; Hydrogen Bonding; Inhibitory Concentration 50; Models, Molecular; Receptors, Estrogen; Structure-Activity Relationship | 2017 |